Robert W. Buckheit : rechercher sur Z-Library

Le plus grand référentiel d'articles scientifiques au monde. 70,000,000+ d'articles gratuitement.

Don't use scam websites

Livres
Articles (165)
Les plus populaires
Liste
- Liste
- Tableau

1

Antiviral activity of hop constituents against a series of DNA and RNA viruses

Victor E Buckwold, Richard J.H Wilson, Aysegul Nalca, Brigitte B Beer, Thomas G Voss, Jim A Turpin, Robert W Buckheit III, Jiayi Wei, Michelle Wenzel-Mathers, Eve M Walton, Robert J Smith, Melanie Pal

Journal:

Antiviral Research

Année:

2004

Langue:

english

Fichier:

PDF, 83 KB

english, 2004

2

Antireplicative and anticytopathic activities of prostratin, a non-tumor-promoting phorbol ester, against human immunodeficiency virus (HIV)

Robert J Gulakowski, James B McMahon, Robert W Buckheit Jr., Kirk R Gustafson, Michael R Boyd

Journal:

Antiviral Research

Année:

1997

Langue:

english

Fichier:

PDF, 353 KB

english, 1997

3

HIV inhibitory natural products. Part 7. The calanolides, a novel HIV-inhibitory class of coumarin derivatives from the tropical rainforest tree, Calophyllum lanigerum

Kashman, Yoel, Gustafson, Kirk R., Fuller, Richard W., Cardellina, John H., McMahon, James B., Currens, Michael J., Buckheit, Robert W., Hughes, Stephen H., Cragg, Gordon M., Boyd, Michael R.

Journal:

Journal of Medicinal Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 1.19 MB

english, 1992

4

Replacement of the Metabolically Labile Methyl Esters in the Alkenyldiarylmethane Series of Non-Nucleoside Reverse Transcriptase Inhibitors with Isoxazolone, Isoxazole, Oxazolone, or Cyano Substituents

Deng, Bo-Liang, Hartman, Tracy L., Buckheit,, Robert W., Pannecouque, Christophe, De Clercq, Erik, Cushman, Mark

Journal:

Journal of Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 127 KB

english, 2006

5

A TIBO derivative, R82913, is a potent inhibitor of HIV-1 reverse transcriptase with heteropolymer templates

E. Lucile White, Robert W. Buckheit Jr, Larry J. Ross, Julie M. Germany, Koen Andries, Rudi Pauwels, Paul A.J. Janssen, William M. Shannon, Michael A. Chirigos

Journal:

Antiviral Research

Année:

1991

Langue:

english

Fichier:

PDF, 538 KB

english, 1991

6

The implications of viral reservoirs on the elite control of HIV-1 infection

Buckheit III, Robert W., Salgado, Maria, Martins, Karen O., Blankson, Joel N.

Journal:

Cellular and Molecular Life Sciences

Année:

2013

Langue:

english

Fichier:

PDF, 563 KB

english, 2013

7

Correlation of Anti-HIV Activity with Anion Spacing in a Series of Cosalane Analogues with Extended Polycarboxylate Pharmacophores

Santhosh, Kalpathy C., Paul, Gitendra C., De Clercq, Erik, Pannecouque, Christophe, Witvrouw, Myriam, Loftus, Tracy L., Turpin, Jim A., Buckheit,, Robert W., Cushman, Mark

Journal:

Journal of Medicinal Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 257 KB

english, 2001

8

More…? Less…? Just Right…? The Role of Perceived Volume in Gel and Film Perceptibility During Intercourse, and its Impact on Product Preference

Morrow, Kathleen M., Rosen, Rochelle K., Vargas, Sara, Katz, David, Joseph, Fava, Kojic, Erna M., Friend, David, Rohan, Lisa, Ham, Anthony, Buckheit, Robert

Journal:

AIDS Research and Human Retroviruses

Année:

2014

Langue:

english

Fichier:

PDF, 61 KB

english, 2014

9

Novel 5′-Norcarbocyclic Pyrimidine Derivatives as Antibacterial Agents

Khandazhinskaya, Anastasia, Alexandrova, Liudmila, Matyugina, Elena, Solyev, Pavel, Efremenkova, Olga, Buckheit, Karen, Wilkinson, Maggie, Buckheit, Robert, Chernousova, Larisa, Smirnova, Tatiana, And

Journal:

Année:

2018

Langue:

english

Fichier:

PDF, 1.60 MB

english, 2018

10

Investigation of 5’-Norcarbocyclic Nucleoside Analogues as Antiprotozoal and Antibacterial Agents

Khandazhinskaya, Anastasia, Matyugina, Elena, Solyev, Pavel, Wilkinson, Maggie, Buckheit, Karen, Buckheit, Robert, Chernousova, Larisa, Smirnova, Tatiana, Andreevskaya, Sofya, Alzahrani, Khalid, Natto

Journal:

Année:

2019

Langue:

english

Fichier:

PDF, 902 KB

english, 2019

11

Synthesis and Biological Activity of 2′-Fluoro-D-arabinofuranosylpyrazolo[3,4-d]pyrimidine Nucleosides

Anita T. Shortnacy-Fowler, Kamal N. Tiwari, John A. Montgomery, Robert W. Buckheit, Jr., John A. Secrist III, Frank Seela

Journal:

Helvetica Chimica Acta

Année:

1999

Langue:

english

Fichier:

PDF, 91 KB

english, 1999

12

ChemInform Abstract: Synthesis and Anti-HIV Activity of Cosalane Analogues with Substituted Benzoic Acid Rings Attached to the Pharmacophore Through Methylene and Amide Linkers.

Jeffrey A. Ruell, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L. Stup, Jim A. Turpin, Robert W. Buckheit Jr., Mark Cushman

Journal:

Année:

1999

Fichier:

PDF, 35 KB

1999

13

ChemInform Abstract: Synthesis and Biological Activity of 2′-Fluoro-D-arabinofuranosylpyrazolo[3,4-d]pyrimidine Nucleosides.

Anita T. Shortnacy-Fowler, Kamal N. Tiwari, John A. Montgomery, Robert W. Buckheit Jr., John A. Secrist III, Frank Seela

Journal:

Année:

2000

Fichier:

PDF, 26 KB

2000

14

ChemInform Abstract: Synthesis of Alkenyldiarylmethane (ADAM) Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors with Non-identical Aromatic Rings.

Guozhang Xu, Tracy L. Hartman, Heather Wargo, Jim A. Turpin, Robert W. Buckheit Jr., Mark Cushman

Journal:

Année:

2002

Fichier:

PDF, 35 KB

2002

15

Development of a combination microbicide gel formulation containing IQP-0528 and tenofovir for the prevention of HIV infection

Anthony S. Ham, Shweta R. Ugaonkar, Lianjun Shi, Karen Watson Buckheit, Howard Lakougna, Umadevi Nagaraja, Garry Gwozdz, Laurie Goldman, Patrick F. Kiser, Robert W. Buckheit Jr.

Journal:

Journal of Pharmaceutical Sciences

Année:

2012

Langue:

english

Fichier:

PDF, 460 KB

english, 2012

16

Optimization of unique, uncharged thioesters as inhibitors of HIV replication

Pratibha Srivastava, Marco Schito, Rasem J. Fattah, Toshiaki Hara, Tracy Hartman, Robert W. Buckheit Jr., Jim A. Turpin, John K. Inman, Ettore Appella

Journal:

Bioorganic & Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 399 KB

english, 2004

17

Synthesis and anti-HIV activity of new alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors (NNRTIs) incorporating benzoxazolone and benzisoxazole rings

Bo-Liang Deng, Matthew D. Cullen, Zhigang Zhou, Tracy L. Hartman, Robert W. Buckheit Jr., Christophe Pannecouque, Erik De Clercq, Phillip E. Fanwick, Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 484 KB

english, 2006

18

Enzymatic triggered release of an HIV-1 entry inhibitor from prostate specific antigen degradable microparticles

Meredith R. Clark, Hyder A. Aliyar, Chang-won Lee, Julie I. Jay, Kavita M. Gupta, Karen M. Watson, Russell J. Stewart, Robert W. Buckheit, Patrick F. Kiser

Journal:

International Journal of Pharmaceutics

Année:

2011

Langue:

english

Fichier:

PDF, 802 KB

english, 2011

19

Synthesis and biological evaluation of an alkenyldiarylmethane (ADAM) which acts as a novel non-nucleoside HIV-1 reverse transcriptase inhibitor

Mark Cushman, Marek Golebiewski, Robert W. Buckheit Jr., Lisa Graham, William G. Rice

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1995

Langue:

english

Fichier:

PDF, 204 KB

english, 1995

20

Inhibition of tubulin polymerization by select alkenyldiarylmethanes

Matthew D. Cullen, Taradas Sarkar, Ernest Hamel, Tracy L. Hartman, Karen M. Watson, Robert W. Buckheit Jr., Christophe Pannecouque, Erik De Clercq, Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 169 KB

english, 2008

21

Investigation of the alkenyldiarylmethane non-nucleoside reverse transcriptase inhibitors as potential cAMP phosphodiesterase-4B2 inhibitors

Matthew D. Cullen, York-Fong Cheung, Miles D. Houslay, Tracy L. Hartman, Karen M. Watson, Robert W. Buckheit Jr., Christophe Pannecouque, Erik De Clercq, Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 136 KB

english, 2008

22

Multivalent binding oligomers inhibit HIV Tat–TAR interaction critical for viral replication

Deyun Wang, Jaclyn Iera, Heather Baker, Priscilla Hogan, Roger Ptak, Lu Yang, Tracy Hartman, Robert W. Buckheit Jr., Alexandre Desjardins, Ao Yang, Pascale Legault, Venkat Yedavalli, Kuan-Teh Jeang, D

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2009

Langue:

english

Fichier:

PDF, 347 KB

english, 2009

23

Synthesis of alkenyldiarylmethanes (ADAMs) containing benzo[d]isoxazole and oxazolidin-2-one rings, a new series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors

Bo-Liang Deng, Yujie Zhao, Tracy L. Hartman, Karen Watson, Robert W. Buckheit Jr., Christophe Pannecouque, Erik De Clercq, Mark Cushman

Journal:

European Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 222 KB

english, 2009

24

Synthesis and anti-HIV activity of a bile acid analog of cosalane

Arunachalam Kannan, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L Hartman, Jim A Turpin, Robert W Buckheit Jr., Mark Cushman

Journal:

Année:

2001

Langue:

english

Fichier:

PDF, 166 KB

english, 2001

25

Identification of optimal anion spacing for anti-HIV activity in a series of cosalane tetracarboxylates

Gitendra C Paul, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L Loftus, Jim A Turpin, Robert W Buckheit Jr., Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2000

Langue:

english

Fichier:

PDF, 285 KB

english, 2000

26

Anti-HIV activity of a series of cosalane amino acid conjugates

Kalpathy C Santhosh, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L Loftus, Jim A Turpin, Robert W Buckheit Jr., Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2000

Langue:

english

Fichier:

PDF, 279 KB

english, 2000

27

In vitro anti-human immunodeficiency virus (HIV) activity of the chromanone derivative, 12-oxocalanolide A, a novel NNRTI

Ze-Qi Xu, Robert W. Buckheit Jr., Tracy L. Stup, Michael T. Flavin, Albert Khilevich, John D. Rizzo, Lin Lin, David E. Zembower

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1998

Langue:

english

Fichier:

PDF, 337 KB

english, 1998

28

Synthesis and anti-HIV activity of cosalane analogues incorporating two dichlorodisalicylmethane pharmacophore fragments

Agustin Casimiro-Garcia, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L Loftus, Jim A Turpin, Robert W Buckheit Jr., Phillip E Fanwick, Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 356 KB

english, 2001

29

Synthesis of substituted diarylmethylenepiperidines (DAMPs), a novel class of anti-HIV agents

Guozhang Xu, Arunachalam Kannan, Tracy L Hartman, Heather Wargo, Karen Watson, Jim A Turpin, Robert W Buckheit Jr., Allison A Johnson, Yves Pommier, Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2002

Langue:

english

Fichier:

PDF, 236 KB

english, 2002

30

Green-to-red photoconvertible fluorescent proteins: tracking cell and protein dynamics on standard wide-field mercury arc-based microscopes

Susan M Baker, Robert W Buckheit, Matthias M Falk

Journal:

BMC Cell Biology

Année:

2010

Langue:

english

Fichier:

PDF, 4.06 MB

english, 2010

31

1-Benzyl derivatives of 5-(arylamino)uracils as anti-HIV-1 and anti-EBV agents

Mikhail S. Novikov, Robert W. Buckheit Jr., Kartik Temburnikar, Anastasia L. Khandazhinskaya, Alexander V. Ivanov, Katherine L. Seley-Radtke

Journal:

Bioorganic & Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 358 KB

english, 2010

32

Synthesis of alkenyldiarylmethane (ADAM) non-Nucleoside HIV-1 reverse transcriptase inhibitors with non-Identical aromatic rings

Guozhang Xu, Tracy L. Hartman, Heather Wargo, Jim A. Turpin, Robert W. Buckheit Jr., Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2002

Langue:

english

Fichier:

PDF, 177 KB

english, 2002

33

Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain

Agustin Casimiro-Garcia, Erik De Clercq, Christophe Pannecouque, Myriam Witvrouw, Tracy L. Stup, Jim A. Turpin, Robert W. Buckheit Jr., Mark Cushman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2000

Langue:

english

Fichier:

PDF, 233 KB

english, 2000

34

Azodicarbonamide inhibits HIV-1 replication by targeting the nucleocapsid protein

Clanton, David, Buckheit, Robert W., Covell, David G., Wallqvist, Anders, McDonnell, Nazli B., DeGuzman, Roberto N., Summers, Michael F., Rice, William G., Turpin, Jim A., Huang, Mingjun

Journal:

Nature Medicine

Année:

1997

Fichier:

PDF, 525 KB

1997

35

5,5-Disubstituted hydantoins: syntheses and anti-HIV activity

Comber, Robert N., Reynolds, Robert C., Friedrich, Joyce D., Manguikian, Roupen A., Buckheit, Robert W., Truss, Jackie W., Shannon, William M., Secrist, John A.

Journal:

Journal of Medicinal Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 774 KB

english, 1992

36

New Alkenyldiarylmethanes with Enhanced Potencies as Anti-HIV Agents Which Act as Non-Nucleoside Reverse Transcriptase Inhibitors

Cushman, Mark, Casimiro-Garcia, Agustin, Hejchman, Elzbieta, Ruell, Jeffrey A., Huang, Mingjun, Schaeffer, Catherine A., Williamson, Karen, Rice, William G., Buckheit, Robert W.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 255 KB

english, 1998

37

Resistance to 1-[(2-Hydroxyethoxy)methyl]-6-(phenylthio)thymine Derivatives Is Generated by Mutations at Multiple Sites in the HIV-1 Reverse Transcriptase

Robert W. Buckheit Jr., Valerie Fliakas-Boltz, Sharon Yeagy-Bargo, Owen Weislow, Douglas L. Mayers, Paul L. Boyer, Stephen H. Hughes, Bai-Chuan Pan, Shih-Hsi Chu, John P. Bader

Journal:

Année:

1995

Fichier:

PDF, 469 KB

1995

38

Vaginal Film Drug Delivery of the Pyrimidinedione IQP-0528 for the Prevention of HIV Infection

Anthony S. Ham, Lisa Cencia Rohan, Ashlee Boczar, Lu Yang, Karen W. Buckheit, Robert W. Buckheit Jr.

Journal:

Pharmaceutical Research

Année:

2012

Langue:

english

Fichier:

PDF, 416 KB

english, 2012

39

Novel sulfonated and phosphonated analogs of distamycin which inhibit the replication of HIV

David J. Clanton, Robert W. Buckheit Jr., Sara J. Terpening, Rebecca Kiser, Nicola Mongelli, Andrea Lombardi Borgia, Robert Schultz, Ven Narayanan, John P. Bader, William G. Rice

Journal:

Antiviral Research

Année:

1995

Langue:

english

Fichier:

PDF, 912 KB

english, 1995

40

Antiviral activity of a phosphorothioate oligonucleotide complementary to human cytomegalovirus RNA when used in combination with antiviral nucleoside analogs

Raana F. Azad, Vickie Brown-Driver, Robert W. Buckheit Jr., Kevin P. Anderson

Journal:

Antiviral Research

Année:

1995

Langue:

english

Fichier:

PDF, 648 KB

english, 1995

41

Comparative anti-HIV evaluation of diverse HIV-1-specific reverse transcriptase inhibitor-resistant virus isolates demonstrates the existence of distinct phenotypic subgroups

Robert W. Buckheit Jr., Valerie Fliakas-Boltz, William Don Decker, Joseph L. Roberson, Tracy L. Stup, Cathi A. Pyle, E.Lucile White, James B. McMahon, Michael J. Currens, Michael R. Boyd, John P. Bade

Journal:

Antiviral Research

Année:

1995

Langue:

english

Fichier:

PDF, 992 KB

english, 1995

42

In vivo drug screening applications of HIV-infected cells cultivated within hollow fibers in two physiologic compartments of mice

Melinda Hollingshead, Joseph Roberson, William Decker, Robert Buckheit Jr., Cindy Elder, Louis Malspeis, Joseph Mayo, Michael Grever

Journal:

Antiviral Research

Année:

1995

Langue:

english

Fichier:

PDF, 880 KB

english, 1995

43

Human immunodeficiency virus type-1 (HIV-1) replication is unaffected by human secretory leukocyte protease inhibitor

Jim A. Turpin, Catherine A. Schaeffer, Ming Bu, Lisa Graham, Robert W. Buckheit Jr., David Clanton, William G. Rice

Journal:

Antiviral Research

Année:

1996

Langue:

english

Fichier:

PDF, 664 KB

english, 1996

44

Development of Anti-Infective Topical Microbicides: 2. Quantifying Inhibition of Virus Transmission in Microbicidal Setting

Karen Watson, Lu Yang, Robert Buckheit Jr.

Journal:

Antiviral Research

Année:

2007

Langue:

english

Fichier:

PDF, 54 KB

english, 2007

45

Development of Anti-Infective Topical Microbicides: 3. Combination Microbicidal Approaches Targeting Multiple Virus Targets or Utilizing Multi-Functional Anti-Infective Agents

Karen Watson, Tracy Hartman, Lu Yang, Robert Buckheit Jr.

Journal:

Antiviral Research

Année:

2007

Langue:

english

Fichier:

PDF, 58 KB

english, 2007

46

Development of Anti-Infective Topical Microbicides: 1. Effects of Seminal and Vaginal Fluids and Other Additives on Viral Infection and Drug Efficacy

Karen Watson, Lu Yang, Robert Buckheit Jr.

Journal:

Antiviral Research

Année:

2007

Langue:

english

Fichier:

PDF, 54 KB

english, 2007

47

Novel Mechanism of Action of Pyrimidinediones Yields Enhanced Sensitivity to Multi-Drug Resistant Virus Strains

Robert W. Buckheit Jr., Lu Yang, Tracy L. Hartman, Karen M. Watson

Journal:

Antiviral Research

Année:

2008

Langue:

english

Fichier:

PDF, 113 KB

english, 2008

48

Development of the Dual-Acting Pyrimidinedione IQP0528 as a Vaginal Topical Anti-HIV Microbicide

Karen M. Watson, Lu Yang, Christa E. Buckheit, Robert W. Buckheit Jr.

Journal:

Antiviral Research

Année:

2008

Langue:

english

Fichier:

PDF, 105 KB

english, 2008

49

Resistance to Pyrimidinedione HIV Inhibitors Requires Multiple Mutations in Reverse Transcriptase, Envelope and Core Proteins

Robert W. Buckheit Jr., Christa E. Buckheit, Robert W. Buckheit III, Karen M. Watson

Journal:

Antiviral Research

Année:

2008

Langue:

english

Fichier:

PDF, 78 KB

english, 2008

50

PG 301029 Inhibits HCV Replication Through a Novel Late Stage Mechanism of Action

Todd B. Parsley, Lu Yang, Robert W. Buckheit Jr.

Journal:

Antiviral Research

Année:

2008

Langue:

english

Fichier:

PDF, 67 KB

english, 2008